Search on: CALCIMIMETIC AGENTS 
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Descriptor English:   Calcimimetic Agents 
Descriptor Spanish:   calcimiméticos 
Descriptor Portuguese:   Calcimiméticos 
Synonyms English:   Agents, Calcimimetic  
Tree Number:   D06.347.230
D27.505.696.399.450.230
Definition English:   Small organic molecules that act as allosteric activators of the calcium sensing receptor (CaSR) in the PARATHYROID GLANDS and other tissues. They lower the threshold for CaSR activation by extracellular calcium ions and diminish PARATHYROID HORMONE (PTH) release from parathyroid cells. 
History Note English:   2011 
Allowable Qualifiers English:  
AD administration & dosage AE adverse effects
AG agonists AN analysis
BL blood CF cerebrospinal fluid
CS chemical synthesis CH chemistry
CL classification EC economics
HI history IM immunology
IP isolation & purification ME metabolism
PK pharmacokinetics PD pharmacology
PO poisoning RE radiation effects
ST standards SD supply & distribution
TU therapeutic use TO toxicity
UR urine  
Record Number:   54038 
Unique Identifier:   D057966 

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